PlumX Metrics
Embed PlumX Metrics

An updated research of glycogen synthase kinase-3β inhibitors: a review

Monatshefte fur Chemie, ISSN: 0026-9247, Vol: 152, Issue: 1, Page: 19-33
2021
  • 4
    Citations
  • 0
    Usage
  • 12
    Captures
  • 0
    Mentions
  • 6
    Social Media
Metric Options:   Counts1 Year3 Year

Metrics Details

  • Citations
    4
    • Citation Indexes
      4
  • Captures
    12
  • Social Media
    6
    • Shares, Likes & Comments
      6
      • Facebook
        6

Review Description

Abstract: Glycogen synthase kinase-3β (GSK-3β) is a highly conserved multifunctional serine/threonine (Ser/Thr) protein kinase widely expressed in many tissues. GSK-3β inhibitors could be used in the treatment of human key diseases, such as cancer, Alzheimer’s disease, Parkinson’s disease, inflammation, type-II diabetes, and so on, due to the multi-role of GSK-3β in the hepatic glycolysis regulation, cell signaling pathways, and phosphorylation of various proteins. Recently, sets of diverse GSK-3β inhibitors have been prepared, and biologically evaluated in vitro and in vivo in different screening models. This review summarizes the latest developments in GSK-3β inhibitors unclosed from 2015 to 2019, including their structure–activity relationship and bioactivity studies. Graphic abstract: [Figure not available: see fulltext.]

Provide Feedback

Have ideas for a new metric? Would you like to see something else here?Let us know