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Synthesis and biology of the rigidified glutamate analogue, trans -2-carboxyazetidine-3-acetic acid ( t -CAA)

Bioorganic & Medicinal Chemistry Letters, ISSN: 0960-894X, Vol: 6, Issue: 21, Page: 2559-2564
1996
  • 28
    Citations
  • 0
    Usage
  • 4
    Captures
  • 0
    Mentions
  • 0
    Social Media
Metric Options:   Counts1 Year3 Year

Metrics Details

  • Citations
    28
    • Citation Indexes
      28
  • Captures
    4

Article Description

Chemical approaches to the (−)- and (+)- trans -2-carboxyazetidine-3-acetic acids (−)- 1 and (+)- 1, and their homologues (−)- 2 and (+)- 2, compounds that represent rigidified analogues of glutamate (glu), are reported together with the complete biological characterization of (+)- 1 ( t -CAA) at the known glu recognition sites. t -CAA was found to be an inhibitor of Na + -dependent glu uptake and to act as a kainate receptor ligand.

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