PlumX Metrics
Embed PlumX Metrics

Cladosporinone, a new viriditoxin derivative from the hypersaline lake derived fungus Cladosporium cladosporioides

Journal of Antibiotics, ISSN: 1881-1469, Vol: 69, Issue: 9, Page: 702-706
2016
  • 24
    Citations
  • 0
    Usage
  • 24
    Captures
  • 0
    Mentions
  • 0
    Social Media
Metric Options:   Counts1 Year3 Year

Metrics Details

Article Description

A new cytotoxic viriditoxin derivative, cladosporinone (1), along with the known viriditoxin (2) and two viriditoxin derivatives (3 and 4) were obtained from the fungus Cladosporium cladosporioides isolated from the sediment of a hypersaline lake in Egypt. The structure of the new compound (1) was determined by 1D and 2D NMR measurements as well as by high-resolution ESIMS and electronic circular dichroism spectroscopy. All isolated compounds were studied for their cytotoxicity against the murine lymphoma cell line L5187Y and for their antibiotic activity against several pathogenic bacteria. Viriditoxin (2) was the most active compound in both bioassays. Compound 1 also exhibited strong cytotoxicity against the murine lymphoma cell line L5187Y with an IC 50 value of 0.88 μm, whereas its antibiotic activity was weak.

Bibliographic Details

Liu, Yang; Kurtán, Tibor; Yun Wang, Chang; Han Lin, Wen; Orfali, Raha; Müller, Werner Eg; Daletos, Georgios; Proksch, Peter

Springer Science and Business Media LLC

Pharmacology, Toxicology and Pharmaceutics

Provide Feedback

Have ideas for a new metric? Would you like to see something else here?Let us know