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Trisubstitution of pyridine through sequential and regioselective palladium cross-coupling reactions affording analogs of known GPR54 antagonists

RSC Advances, ISSN: 2046-2069, Vol: 3, Issue: 26, Page: 10296-10300
2013
  • 10
    Citations
  • 0
    Usage
  • 15
    Captures
  • 0
    Mentions
  • 0
    Social Media
Metric Options:   Counts1 Year3 Year

Metrics Details

  • Citations
    10
    • Citation Indexes
      9
    • Patent Family Citations
      1
      • Patent Families
        1
  • Captures
    15

Article Description

Because of their large spectrum of applications, poly-functionalized pyridines remain an attractive challenge in modern organic chemistry. We describe the poly-functionalization of halopyridines through a series of sequential and regioselective palladium-catalyzed cross-coupling reactions (Suzuki-Miyaura, Sonogashira and Buchwald-Hartwig reactions). This strategy was applied to the synthesis of several analogs of single non-peptidic known GPR54 antagonists. © The Royal Society of Chemistry 2013.

Bibliographic Details

Christelle Doebelin; Patrick Wagner; Martine Schmitt; Frédéric Bihel; Jean Jacques Bourguignon; Isabelle Bertin; Frédéric Simonin

Royal Society of Chemistry (RSC)

Chemistry; Chemical Engineering

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