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Novel synthesis of fused spiro piperidone-cyclopropanes from cyclopropyl amides and electron-deficient alkenes

Organic and Biomolecular Chemistry, ISSN: 1477-0520, Vol: 19, Issue: 14, Page: 3191-3198
2021
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  • Citations
    2
    • Citation Indexes
      2

Article Description

We report here that a series of bridgedO,O-ketal fused spiro piperidone-cyclopropane derivatives3can be constructed with excellent yields and good diastereoselectivity by the one-pot reaction of 1-acylcyclopropanecarboxamides1with electron-deficient alkene2a(EWG = CHO)viathe domino process involving [4 + 2] annulation/intermolecular electrophilic addition/intramolecular cyclization. Furthermore, reactions of1with2b/2c(EWG = CN, COOMe), leading to spiro piperidone-cyclopropane derivatives4or5by base catalyst selection, were also presented.

Bibliographic Details

Han, Xiao-Dan; Peng, Gao-Liang; Wang, Hui-Bin; Wu, Lei; Fu, Jian-Ping; Tang, Zhong-Sheng; Hu, Ju-Wu; Xiong, Wei

Royal Society of Chemistry (RSC)

Biochemistry, Genetics and Molecular Biology; Chemistry

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